Eikozanoidni receptor

Eikozanoidni receptor je integralni membranski protein koji detektuje prisustvo eikozanoidnih signalnih molekula. Većina, mada ne svi, su G protein spregnuti receptori. Primer ne-GPCR receptora koji vezuje eikozanoide je PPAR-γ.[1]

Ovo su poznati humani eikozanoidni GPCR receptori grupisani po tipu eikozanoidnog liganda koji vezuju:[2][3]

Leukotrien uredi

Leukotrieni:

Lipoksin uredi

Lipoksini:

Oksoeikozanoid uredi

Oksoeikozanoid:[4]

Prostanoid uredi

Prostanoidi:

Reference uredi

  1. DuBois RN, Gupta R, Brockman J, Reddy BS, Krakow SL, Lazar MA (1998). „The nuclear eicosanoid receptor, PPAR-γ, is aberrantly expressed in colonic cancers”. Carcinogenesis 19 (1): 49–53. DOI:10.1093/carcin/19.1.49. PMID 9472692. 
  2. Coleman RA, Smith WL, Narumiya S (1994). „International Union of Pharmacology classification of prostanoid receptors: properties, distribution, and structure of the receptors and their subtypes”. Pharmacol. Rev. 46 (2): 205–29. PMID 7938166. 
  3. Brink C, Dahlén SE, Drazen J, Evans JF, Hay DW, Nicosia S, Serhan CN, Shimizu T, Yokomizo T (2003). „International Union of Pharmacology XXXVII. Nomenclature for leukotriene and lipoxin receptors”. Pharmacol. Rev. 55 (1): 195–227. DOI:10.1124/pr.55.1.8. PMID 12615958. 
  4. Brink C, Dahlén SE, Drazen J, Evans JF, Hay DW, Rovati GE, Serhan CN, Shimizu T, Yokomizo T (2004). „International Union of Pharmacology XLIV. Nomenclature for the oxoeicosanoid receptor”. Pharmacol. Rev. 56 (1): 149–57. DOI:10.1124/pr.56.1.4. PMID 15001665. 

Spoljašnje veze uredi